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Venlafaxine CAS:93413-69-5

Venlafaxine bụ ọgwụ na-ebelata nchekasị nke klaasị serotonin na norepinephrine reuptake inhibitor (SNRI). Wyeth mepụtara ọgwụ a na 19Chemicalbook93 ma ugbu a Pfizer na-ere ya. A kwadoro ọgwụ a maka ọgwụgwọ nke nnukwu nsogbu ịda mbà n'obi (MDD), nsogbu nchekasị zuru oke (GAD), na ịda mbà n'obi nke metụtara nchekasị.


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Ngwa na Mmetụta

Venlafaxine nwere ike igbochi nlọghachi nke NA na 5-HT, ma gbochiekwa dopamine ịmaliteghachi ọzọ. In vitro mgbochi nke ndị na-anabata cholinergic, ndị na-anabata histamine α Ndị na-anabata ha abụọ enweghị njikọ. Ntinye afọ dị mma, a na-emekwa ka Chemicalbook dị na imeju site na cytochrome P45011D6 ma na-ewepụta ya site na mmamịrị. T1/2 nke metabolites ndị bụ isi na-arụ ọrụ dị site na awa 5 ruo 11. Mgbe izu atọ gachara, e ruru njupụta ọnọdụ kwụsiri ike. Ejiri ya maka ọgwụgwọ nke ịda mbà n'obi.

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Ozi Mgbakwunye:

Ihe mejupụtara ya C17H27NO2
Nnwale 99%
Ọdịdị Ntụ ntụ ọcha
Nọmba CAS 93413-69-5
Nkwakọ ngwaahịa 25KG
Ndụ nchekwa afọ 2
Nchekwa Debe n'ebe dị jụụ ma kpọọ nkụ
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