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Clascoterone CAS:19608-29-8 Onye Na-eweta Ngwaahịa
Clascoterone bụ ọgwụ mgbochi androgen receptor nke Cassiopea (ụlọ ọrụ Cosmo Pharmaceuticals) mepụtara dị ka ude na ngwọta maka nsogbu akpụkpọ ahụ dabere na androgen, gụnyere alopecia androgenic na acne vulgaris. Ọ bụ ezie na amaghị kpọmkwem usoro clascoterone si arụ ọrụ maka ọgwụgwọ acne vulgaris n'elu, a kwenyere na ọgwụ ahụ na-asọmpi na androgen dihydrotestosterone maka ijikọ na androgen receptors na sebaceous gland na follicles ntutu iji belata mgbaàmà dị mkpa maka mmepe nke acne.
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Pitavastatin CAS:147511-69-1 Onye Na-eweta Ngwaahịa
Pitavastatin bụ ihe na-egbochi HMG-CoA reductase nke na-akwalite usoro mbụ nke mmepụta cholesterol. Ọ na-adị ka ntụ ntụ na-enweghị isi ma na-acha ọcha ruo na-acha odo odo. Ọ na-arụ ọrụ site n'ibelata ọkwa nke ụfọdụ ihe abụba dị ka cholesterol n'ahụ. Ya mere, a na-egosi ya karịsịa maka ọgwụgwọ hypercholesterolemia na maka igbochi ọrịa obi. Ọ bụghị naanị na ọ nwere ike ibelata cholesterol dị elu na triglyceride n'ime ụfọdụ ndị ọrịa, kamakwa ọ nwere ike ịbawanye ọdịnaya nke lipoprotein dị elu (HDL), ọkwa cholesterol "dị mma". A ga-ejikarị ya na nri kwesịrị ekwesị.
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Teduglutide CAS:197922-42-2 Onye Na-eweta Ngwaahịa
Teduglutide (a makwaara dịka ALX-0600) bụ ihe atụ GLP-2 ebe ejiri glycine dochie alanine na ọnọdụ nke abụọ site na N-terminus, si otú a na-egbochi mbibi site na DPP-4. Teduglutide nwere njikọ yiri nke ahụ, ike agonist, na arụmọrụ agonist dị ka GLP-2 na nnwale na oke GLP-2 receptor. Ntinye teduglutide nye oke nyere mmụba dị ukwuu na ibu obere eriri afọ na mmụba na elu nke eriri afọ villi. E ji usoro peptide siri ike kwadebe Teduglutide.
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Malic Acid CAS:6915-15-7 Onye Na-eweta Ngwaahịa
Malic acid bụ 2-hydroxydicarboxylic acid nke bụ succinic acid nke otu hydrogen jikọtara na carbon na-anọchi otu hydroxy group. Ọ nwere ọrụ dị ka ihe na-achịkwa acidity nri na metabolite bụ isi. Ọ bụ 2-hydroxydicarboxylic acid na C4-dicarboxylic acid. Ọ na-enweta site na succinic acid. Ọ bụ conjugate acid nke malate(2-) na malate.
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Gabapentin CAS:60142-96-3 Onye Na-eweta Ngwaahịa
Gabapentin bụ isi ihe na-egbochi akwara ozi nke na-arụ ọrụ site na ijikọ na ndị na-anabata GABA dị na eriri azụ. Gabapentin bụ γ-aminobutyric acid (GABA) analog nke na-arụ ọrụ dị ka anticonvulsant nwere mmetụta mgbu a nwapụtara na ọtụtụ ọrịa mgbu neuropathic dịka Complex Regional Pain Syndrome type one (CRPS 1).
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Paracetamol CAS:103-90-2 Onye Na-eweta Ngwaahịa
Paracetamol bụ otu n'ime phenols nke bụ 4-aminophenol nke otu acetyl dochie otu n'ime hydrogen ndị dị na otu amino. Ọ nwere ọrụ dị ka ihe mgbochi cyclooxygenase 2, ihe mgbochi cyclooxygenase 1, ihe mgbu na-abụghị narcotic, ihe mgbochi antipyretic, ọgwụ mgbochi mkpali na-abụghị steroidal, ihe mgbochi cyclooxygenase 3, ihe na-egbochi xenobiotic, ihe na-emebi gburugburu ebe obibi, ihe na-eme ka ọbara mmadụ dị n'ọbara, ihe na-eme ka hepatotoxic pụta, ihe na-akpali ferroptosis na ihe na-echebe geroprotector. Ọ bụ otu phenols na onye otu acetamides. Ọ nwere njikọ ọrụ na 4-aminophenol.
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Calcium Aspartate CAS:10389-09-0 Onye Na-eweta Ngwaahịa
Calcium Aspartatebụ otu n'ime mineral kachasị baa ụba n'ahụ ma bụrụkwa ihe dị mkpa ná ndụ anyị. Na-enweghị ya, ụmụ mmadụ agaghị enwe ike ịnọgide na-enwe ọkpụkpụ na ezé siri ike. Ihe dị ka 99% nke calcium dị n'ahụ dị n'ebe abụọ a. Na mgbakwunye, calcium na-enyere obi, akwara, akwara na sistemụ ndị ọzọ nke ahụ aka ịrụ ọrụ nke ọma. Ọ nwere nhazi kemịkalụ kwụsiri ike, ezigbo mmiri na-agbaze na oke nnabata. Ọ bụ nke ọgbọ kachasị ọhụrụ nke ihe na-eme ka calcium sie ike.
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L-Carnitine L-Tartrate CAS:36687-82-8 Onye Na-eweta Ngwaahịa
L-carnitine bụ ihe sitere n'okike nke amino acid nke a na-eji dị ka ihe mgbakwunye maka mbelata ibu. L-carnitine-L-tartrate (LCLT) bụ nnu nke L-carnitine nwere tartaric acid. LCLT nwere ike ime ka kemịkalụ na ihe ndị na-egbochi antioxidant dị ike..
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Miconazole CAS:22916-47-8 Onye Na-eweta Ngwaahịa
Miconazole (Monistat) bụ ọgwụ nje imidazole nke a na-eji agwọ ọrịa akpụkpọ ahụ na ọrịa akpụkpọ ahụ na-efe efe nke Candida, dị ka vaginitis. Ọ na-esi n'elu akpụkpọ ahụ ma ọ bụ akpụkpọ ahụ mucous apụta ntakịrị. Enwere ike ime ka akpụkpọ ahụ na akpụkpọ ahụ na akpụkpọ ahụ mucous apụta site n'iji ya n'elu; a kọọla isi ọwụwa, urticaria, na afọ mgbu na ọgwụgwọ maka vaginitis.
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Nnu Pyrroloquinoline Quinone Disodium CAS:122628-50-6
Nnu Pyrroloquinoline quinone disodium bụ ngwakọta quinone na-agbaze mmiri nke nwere ikike antioxidant siri ike. Ngwaahịa a bụ ntụ ntụ agba aja aja na-acha ọbara ọbara. A na-ekewapụ ya na ọdịbendị nke nje bacteria methylotrophic na anụ ahụ nke anụmanụ. Nri a dị mkpa dị mkpa maka anụmanụ, na-arụ ọrụ dị mkpa n'ịkwalite ọrụ ahụ ji alụso ọrịa ọgụ.
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Citrulline CAS:372-75-8 Onye Na-eweta Ngwaahịa
Citrulline bụ L-enantiomer nke citrulline. Ọ nwere ọrụ dịka ihe mgbochi EC 1.14.13.39 (nitric oxide synthase), ihe na-egbochi ihe, ihe na-edozi ahụ, ihe na-edozi ahụ, ihe na-edozi ahụ, ihe na-edozi ahụ mmadụ, ihe na-eme ka Escherichia coli dị n'ime, ihe na-eme ka Saccharomyces cerevisiae dị n'ime na ihe na-eme ka òké dị n'ime. Ọ bụ enantiomer nke D-citrulline. Ọ bụ tautomer nke L-citrulline zwitterion.
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L-Arginine Alfa-Ketoglutarate (2: 1) Dihydrate CAS: 5256-76-8
L-Arginine Alfa-Ketoglutarate (2: 1) Dihydratebụ ngwaahịa ọgwụ nke so n'òtù ọgwụ eji agwọ hyperlipidemia. Nhazi nke ọgwụ a nwere molekul arginine abụọ ejikọtara na atọm oxygen. Ọ bụ kristal siri ike nke nwere dayameta nkezi nke 0.3 μm na nkesa nha nke ihe dị n'etiti 0.05 na 1.5 μm.
