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Isi Hydrocortisone CAS:50-23-7 Onye Na-emepụta Ihe
Hydrocortisone, 11β,17,21-trihydroxypregn-4-ene-3,20-dione, bụ GCin bụ isi mmadụ. N'agbanyeghị ọtụtụ GCs e ji aka mee, hydrocortisone, esters ya, na nnu ya ka bụ isi ihe dị mkpa n'ọgwụgwọ steroid adrenocortical nke oge a na ọkọlọtọ maka iji tụnyere GCs na MCs ndị ọzọ niile. A na-eji ya maka ihe ngosi niile a kpọtụrụ aha na mbụ.
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Orlistat CAS:96829-58-2 Onye Na-eweta Ngwaahịa
Orlistat bụ ọgwụ mgbochi lipase nke na-egbochi nri. E wepụtara Orlistat na UK dị ka Xenical maka ọgwụgwọ ogologo oge nke oke ibu, ọkachasị na nri nwere obere kalori. Orlistat bụ ọgwụ sitere na hypolipaemic lipstatin eke (site na Streptomyces toxyfncini) a na-enweta site na hydrogenation nke lipstatine ma ọ bụ site na ọtụtụ ụzọ sịntetik dị iche iche gụnyere ọtụtụ nzọụkwụ site na (S) - rnalic acid.
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L-Homoarginine Monohydrochloride CAS:1483-01-8 Onye Na-eweta Ngwaahịa
L-Homoarginine bụ ihe na-egbochi phosphatases alkaline nke na-anaghị asọmpi ma na-egbochi akụkụ ahụ. Amino acid a na-adịghị mkpa na-egbochi phosphatases alkaline ọkpụkpụ mmadụ na imeju mana ọ nweghị mmetụta ọ bụla na isoenzymes nke placental ma ọ bụ eriri afọ. Ọgwụgwọ tupu L-homoarginine na-egbu oge uto etuto ahụ na vivo na ụdị C3H/He osteosarcoma murine. Ọ na-egbochikwa uto pancreatic nke nwere protein dị elu na mmepụta enzyme na oke bile-pancreatic juice-diverted, ihe nlereanya maka mkpali nke mmepụta enzyme pancreatic na hypercholecystokininemia..
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Escitalopram Oxalate CAS:219861-08-2
Escitalopram oxalate bụ metabolite S-isomer nke citalopram na akụkụ bụ isi nke ọrụ ọgwụ ya. Aha kemịkalụ ya bụ (S) -1- [3- (dimethylamino) propyl] -1- (Chemicalbook4-fluorophenyl) -1,3-dihydroisobenzofuran 5-acetonitrile oxalate, Ọ bụ ihe na-egbochi serotonin reuptake, Ọ nwere mmetụta ọgwụgwọ dị mma na ma endogenous na non-endogenous depression.
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Glutathione Ebelatara CAS:70-18-8 Onye Na-eweta Ngwaahịa
Glutathione (GSH) bụ tripeptide (γ-glutamylcysteinylglycine) nke a na-ekesa n'ọtụtụ ebe n'osisi na anụmanụ. GSH na-eje ozi dị ka ihe mgbakwunye nucleophilic na glutathione transferases na mwepụ nke xenobiotics ma bụrụ ihe dị mkpa nye onye na-enye electron na glutathione peroxidases na mbelata nke hydroperoxides. GSH na-etinyekwa aka na njem amino acid na mmezi nke ọkwa mbelata protein sulfhydryl. Ọnụọgụ nke GSH sitere na obere micromolar na plasma ruo ọtụtụ millimolar na anụ ahụ dịka imeju.
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Cysteine CAS:52-90-4 Onye Na-eweta Ngwaahịa
L-Cysteine bụ otu n'ime amino asịd iri abụọ sitere n'okike, e wezụga methionine, naanị ya nwere sọlfọ. Ọ bụ amino asịd nke na-adịghị mkpa nke nwere thiol nke a na-eme ka ọ ghọọ Cystine. Ọ bụ amino asịd nke na-adịghị mkpa nke nwere sọlfọ n'ime mmadụ, nke metụtara cystine, Cysteine dị mkpa maka njikọ protein, iwepụ nsị, na ọrụ metabolic dị iche iche. A na-ahụ Cysteine na beta-keratin, protein bụ isi dị na mbọ, akpụkpọ ahụ, na ntutu isi, ọ dịkwa mkpa na mmepụta collagen, yana ịgbatị akpụkpọ ahụ na udidi ya.
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Asịd enweghị Coenzyme A CAS:85-61-0
Asịd enweghị Coenzyme Abụ ihe dị mkpa na-arụ ọrụ dị ka ihe na-ebu otu acyl na otu carbonyl na-eme ka carbonyl rụọ ọrụ maka usoro citric acid na metabolism abụba. Ihe dị ka 4% nke enzymes sel na-eji CoA dị ka ihe ndabere. A na-emepụta ya site na pantothenic acid na usoro nzọụkwụ ise nke chọrọ ATP. Achọpụtala nzọụkwụ pantothenate kinase nke ụzọ biosynthetic CoA dị ka ihe mgbaru ọsọ maka mmepe nke ogige nje bacteria.
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Idebenone CAS:58186-27-9 Onye Na-eweta Ngwaahịa
Idebenone bụ ihe mejupụtara organic nke ezinụlọ quinone, nke yiri coenzyme Q-10. Ọ bụ ụdị ọgwụ Takeda Pharmaceutical Company mepụtara maka ọgwụgwọ ọrịa Alzheimer na ụfọdụ nkwarụ ọgụgụ isi ndị ọzọ. Agbanyeghị, ihe ndị a adịchaghị mma metụtara ihe ngosi a. A na-ejikwa ya ugbu a maka ọgwụgwọ Friedreich's ataxia yana mmetụta dị mma na hypertrophy obi na ọrụ akwara ozi.
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Tetracaine Hydrochloride CAS:136-47-0 Onye Na-emepụta Ihe
Tetracaine hydrochloride bụ benzoate ester. Ọ bụ ọgwụ mgbu mpaghara dị ike nke ụdị ester nke a na-eji eme ihe maka anesthesia elu na spinal. Tetracaine hydrochloride bụ ọgwụ mgbu mpaghara yana ihe ester sitere na p-amino benzoic acid. Ọ na-arụ ọrụ site na igbochi ntinye nke ion sodium n'ime mkpụrụ ndụ akwara ma bụrụ otu n'ime ọgwụ mgbu a na-ejikarị eme ihe.
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Leucine CAS:61-90-5 Onye Na-eweta Ngwaahịa
Leucine bụ otu n'ime amino asịd asatọ dị mkpa, ọ bụkwa nke amino asịd aliphatic dị n'ime ụdị protein iri abụọ. A na-akpọ L-leucine na L-isoleucine na L-valine amino asịd atọ nwere alaka. L-leucineLeucine na D-leucine bụ enantiomers. Ọ bụ kristal hexahedral ọcha na-egbuke egbuke ma ọ bụ ntụ kristal ọcha na okpomọkụ ụlọ, enweghị isi, ọ na-ewe ntakịrị ilu. N'ihu hydrocarbons, ọ kwụsiri ike na acid mineral mmiri. A na-agbaze kwa gram na mmiri 40ml na ihe dị ka 100ml acetic acid. Ọ na-agbaze ntakịrị na ethanol ma ọ bụ ether, gbazee na formic acid, gwakọtara hydrochloric acid, ngwọta nke alkali hydroxides na ngwọta nke carbonates.
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Guanidinopropionic Acid CAS:353-09-3 Onye Na-eweta Ngwaahịa
Asịd Guanidinopropionic bụ kristal ọcha nke na-agbaze n'ime mmiri ma bụrụkwa ihe yiri creatine. Asịd Guanidinopropionic bụ ụdị amino acid sitere na ya. Ọ bụ ihe dị mkpa na kemịkalụ ma dịkwa n'etiti. Ọ dị n'ime ọbara, ụbụrụ, imeju, akụrụ na mmamịrị nke anụmanụ.
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Olmesartan CAS:144689-24-7 Onye Na-eweta Ngwaahịa
Olmesartan medoxomil,phenyl]phenyl]methyl]imidazole-4-carboxylate (Benicar, Olmetec) na-eji usoro tetrazolering dị ka sistemụ acidic ya, nke na-esonye na njikọ nke ndị na-anabata ihe. Mgbe e nyere onye ọrịa, ọgwụ a na-eme ka ọ rụọ ọrụ ngwa ngwa ma zuru oke site na ester hydrolysis nke medoxomil mgbe a na-amịkọrọ ya site na eriri afọ. Olmesartan bụ biphenylyltetrazole. Ọ nwere ọrụ dị ka ihe na-egbochi ọbara mgbali elu na ihe na-egbochi ndị na-anabata ihe angiotensin.
